Abstract
Organic compounds containing the thiazolinone ring are of increasing interest due to their bactericidal, pesticidal, anticonvulsant, antiinflammatory, antithyroidal and antimicrobial activities. A rapid microwave-assisted synthesis thiazolinone derivatives is described. The 3-(1H-benzo[d]imidazol-2-yl)-2-substituted phenyl thiazolidin-4-one were identified by IR, 1H NMR, elemental analyses. The target compounds were performed in a shorter reaction time compared to conventional heating methods.
Get full access to this article
View all access options for this article.
References
1.
Nawrocka W.
,
Sztuba B.
,
Kowalska M.W.
,
Liszkiewicz H.
,
Wietrzyk J.
,
Nasulewicz A.
,
Pelczyńska M.
, and
Opolski A.
, Il Farmaco , 2002 , 57 , 101 .
2.
Valdez J.
,
Cedillo R.
,
Hernández-Campos A.
,
Yépez L.
,
Hernández-Luis F.
,
Navarrete-Vázquez G.
,
Tapia A.
,
Cortés R.
,
Hernández M.
, and
Castillo R.
, Bioorg. Med. Chem. Lett. , 2002 , 12 , 2221 .
3.
Li Y.F.
,
Wang G.F.
,
He P.L.
,
Huang W.G.
,
Zhu F.H.
,
Gao H.Y.
,
Tang W.
,
Luo Y.
,
Feng C.L.
,
Shi L.P.
,
Ren Y.D.
,
Lu W.
, and
Zuo J.P.
, J. Med. Chem. , 2006 , 49 , 4790 .
4.
El-masry A.H.
,
Fahmy H.H.
, and
Ali Abdelwahed S.H.
, Molecules , 2000 , 5 , 1429 .
5.
Rogers S.A.
,
Huigens R.W.
III
, and
Melander C.
, J. Am. Chem. Soc. , 2009 , 131 , 9868 .
6.
Chen H.
,
Jiao L.
,
Guo Z.
,
Li X.
,
Ba C.
, and
Zhang J.
, Carbohydr. Res. , 2008 343 , 3015 .
7.
Vicini P.
,
Geronikaki A.
,
Incerti M.
,
Zani F.
,
Deardenc J.
, and
Hewitt M.
, Bioorg. Med. Chem. , 2008 , 16 , 3714 .
8.
Navarrete-Vázquez G.
,
Cedillo R.
,
Hernández-Camposa A.
,
Yépezb L.
,
Hernández-Luisa F.
,
Valdeza J.
,
Moralesb R.
,
Cortésc R.
,
Hernándezc M.
, and
Castilloa R.
, Bioorg. Med. Chem. Lett. , 2001 , 11 , 187 .
9.
Navarrete-Vázquez G.
,
Rojano-Vilchis M.M.
,
Yépez-Mulia L.
,
Meléndez V.
,
Gerena L.
,
Hernández-Campos A.
,
Castillo R.
, and
Hernández-Luis F.
, Eur. J. Med. Chem. , 2006 , 41 , 135 .
10.
Rahman V.P.
,
Mukhtar S.
,
Ansari W.H.
,
Lemiere G.
, Eur. J. Med. Chem. , 2005 , 40 , 173 .
11.
Hu J.
,
Sun J.
,
Zhou T.
, and
Xu Y.
, J. Chem. Res. , 2011 , 35 , 442
12.
Hu J.
,
Wang J.
,
Zhou T.
, and
Xu Y.
, J. Chem. Res. , 35 , 525 .
